
AZD3759 hydrochloride
CAS No. 1626387-81-2
AZD3759 hydrochloride ( —— )
产品货号. M18097 CAS No. 1626387-81-2
AZD3759(盐酸盐)是一种有效的、口服活性的、中枢神经系统渗透性 EGFR 抑制剂。
纯度: >98% (HPLC)






规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥405 | 有现货 |
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5MG | ¥551 | 有现货 |
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10MG | ¥794 | 有现货 |
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25MG | ¥1369 | 有现货 |
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50MG | ¥2414 | 有现货 |
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100MG | ¥3977 | 有现货 |
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500MG | ¥9072 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称AZD3759 hydrochloride
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述AZD3759(盐酸盐)是一种有效的、口服活性的、中枢神经系统渗透性 EGFR 抑制剂。
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产品描述AZD3759 (hydrochloride) is an effective, orally active and central nervous system-penetrant?EGFR?inhibitor. At Km?ATP concentrations, the?IC50s are 0.2/0.3/0.2 nM for EGFR (L858R)/EGFR (wt)/EGFR (exon 19Del).
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体外实验——
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体内实验——
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同义词——
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通路Others
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靶点Other Targets
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受体EGFR (exon 19De)| EGFR (L858R)| EGFR (wt)
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研究领域——
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适应症——
化学信息
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CAS Number1626387-81-2
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分子量496.36
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分子式C22H24Cl2FN5O3
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纯度>98% (HPLC)
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溶解度——
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SMILESC[C@@H]1CN(CCN1C(=O)OC2=C(C=C3C(=C2)C(=NC=N3)NC4=C(C(=CC=C4)Cl)F)OC)C.Cl
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Zeng Q, et al. J Med Chem. 2015 Oct 22;58(20):8200-15.
产品手册




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