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AZD3759 hydrochloride

CAS No. 1626387-81-2

AZD3759 hydrochloride ( —— )

产品货号. M18097 CAS No. 1626387-81-2

AZD3759(盐酸盐)是一种有效的、口服活性的、中枢神经系统渗透性 EGFR 抑制剂。

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
2MG ¥405 有现货
5MG ¥551 有现货
10MG ¥794 有现货
25MG ¥1369 有现货
50MG ¥2414 有现货
100MG ¥3977 有现货
500MG ¥9072 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    AZD3759 hydrochloride
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    AZD3759(盐酸盐)是一种有效的、口服活性的、中枢神经系统渗透性 EGFR 抑制剂。
  • 产品描述
    AZD3759 (hydrochloride) is an effective, orally active and central nervous system-penetrant?EGFR?inhibitor. At Km?ATP concentrations, the?IC50s are 0.2/0.3/0.2 nM for EGFR (L858R)/EGFR (wt)/EGFR (exon 19Del).
  • 体外实验
    ——
  • 体内实验
    ——
  • 同义词
    ——
  • 通路
    Others
  • 靶点
    Other Targets
  • 受体
    EGFR (exon 19De)| EGFR (L858R)| EGFR (wt)
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    1626387-81-2
  • 分子量
    496.36
  • 分子式
    C22H24Cl2FN5O3
  • 纯度
    >98% (HPLC)
  • 溶解度
    ——
  • SMILES
    C[C@@H]1CN(CCN1C(=O)OC2=C(C=C3C(=C2)C(=NC=N3)NC4=C(C(=CC=C4)Cl)F)OC)C.Cl
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1. Zeng Q, et al. J Med Chem. 2015 Oct 22;58(20):8200-15.
产品手册
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